1. APIs
  2. Ulipristal Acetate
  3. ULIPA Metabolites
  4. Mono-N-demethylated Ulipristal Acetate

Mono-N-demethylated Ulipristal Acetate

Structure

Notes

Also known as metabolite PGL4002. Pharmacologically active. Binds to human plasma proteins extensively at 96.5%. Most likely mediated by CYP3A4.

References

  1. Product Monograph: Fibristal, 5 mg ulipristal acetate tablet. Allergan Pharma Co. Nov. 23, 2016. (View all citations for this reference)
  2. 30 mg ulipristal acetate tablet for emergency contraception. Laboratoire HRA Pharma, Distributed by: Actavis Specialty Pharmaceuticals Co. January 22, 2015. (View all citations for this reference)