Citations for: Sitruk-Ware, R.; Small, M.; Kumar, N.; Tsong, Y.-Y.; Sundaram, K.; Jackanicz, T., Nestorone®: clinical applications for contraception and HRT. Steroids 2003, 68 (10-13), 907-913.

Entry Type
Name
Value
Parent Entry
Pharmacology Data Field
Androgen Receptor Activity
Reported as weakly effective to effective agonist.
Medroxy­progesterone Acetate (API)
Pharmacology Data Field
Androgen Receptor Activity
No activity
Nestorone (API)
Pharmacology Data Field
Estrogen Receptor Activity
Antagonist
Nestorone (API)
Pharmacology Data Field
Serum Protein Binding
Binds to albumin. Does not bind to SHBG.
Nestorone (API)
Pharmacology Data Field
Androgen Receptor Activity
Antagonist (40% of CPA, the most potent anti-androgenic progestin)
Dienogest (API)